SCHEMBL15501094

SCHEMBL15501094

C=NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](CCCCC/C=C\[C@@H]1C[C@@H]1C(=O)OCC)NC(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC4 P56524 2/20 0.33
ITGB3 P05106 7/20 0.32
ITGA2B P08514 7/20 0.32
CTSL P07711 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
TGM2 P21980 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6124828 0.90 HDAC1 (0.35) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL7941871 0.90 HDAC1 (0.35) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL13435766 0.81 ATM (0.32)
SCHEMBL13071444 0.80 ITGB3 (0.37) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL8203250 0.80 F2 (0.41) HDAC1HDAC4ITGB3ITGA2BCTSL
SCHEMBL6383995 0.80 ITGB3 (0.39) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL13435882 0.80 F2 (0.40) ITGB3ITGA2B
SCHEMBL14216849 0.78 HDAC1 (0.32) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL13071545 0.77 HDAC1 (0.39) HDAC1HDAC8HDAC4ITGB3ITGA2B
SCHEMBL10166392 0.77 HDAC1 (0.35) HDAC1HDAC8HDAC4ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323981-B1 PROCESS FOR THE PREPARATION OF A MACROCYCLE HOFFMANN LA ROCHE (CH) 2014-03-12 EP disclosed