SCHEMBL1551650

SCHEMBL1551650

Cc1cnc2cc([N+](=O)[O-])ccc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.50
HTT P42858 3/20 0.50
ALDH1A1 P00352 5/20 0.49
TXNRD1 Q16881 1/20 0.49
TXNRD3 Q86VQ6 1/20 0.49
TXNRD2 Q9NNW7 1/20 0.49
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
CYP1A2 P05177 1/20 0.47
MAPT P10636 4/20 0.46
CYP3A4 P08684 2/20 0.46
NAMPT P43490 1/20 0.46
XDH P47989 1/20 0.46
TDP1 Q9NUW8 2/20 0.46
TSHR P16473 1/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
GUCY1B2 O75343 1/20 0.46
GUCY1A2 P33402 1/20 0.46
GUCY1A1 Q02108 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12814503 0.93 SMN1; SMN2 (0.50) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL3720824 0.81 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1TXNRD1TXNRD3TXNRD2
SCHEMBL30891041 0.80 ALDH1A1 (0.49) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL3567491 0.80 ALDH1A1 (0.49) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL3563953 0.80 RAB9A (0.52) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL30891215 0.80 RAB9A (0.52) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL1770090 0.79 SMN1; SMN2 (0.56) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL11263318 0.78 ALDH1A1 (0.44) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL7307217 0.78 ALDH1A1 (0.47) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3
SCHEMBL1207982 0.78 ALDH1A1 (0.57) SMN1; SMN2HTTALDH1A1TXNRD1TXNRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250282748-A1 SUBSTITUTED OXOPYRIDINE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2025-09-11 US disclosed
CN-113292539-B Substituted oxopyridine derivatives 拜耳制药股份公司 2023-12-22 CN disclosed
CN-116410146-A One-step process for converting polyols to nitrogen-containing heterocycles using heterogeneous metal catalysts 浙江大学 2023-07-11 CN disclosed
US-20230024752-A1 SUBSTITUTED OXOPYRIDINE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2023-01-26 US disclosed
CN-113087674-B Method for synthesizing quinoxaline compound under catalysis of visible light induced photosensitizer 河南大学 2022-06-17 CN disclosed
US-11180471-B2 Substituted oxopyridine derivatives BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-11-23 US disclosed
CN-113292539-A Substituted oxopyridine derivatives 拜耳制药股份公司 2021-08-24 CN disclosed
CN-108026072-B Substituted oxopyridine derivatives 拜耳制药股份公司 2021-08-17 CN disclosed
CN-113087674-A Method for synthesizing quinoxaline compound under visible light induced iron catalysis condition 河南大学 2021-07-09 CN disclosed
EP-3319956-B1 SUBSTITUTED OXOPYRIDINE DERIVATIVES Bayer Pharma AG (DE) 2021-01-06 EP disclosed
US-5204347-A Reduction in intraocular pressure; increase renal flow; alteration in the rate of fluid transport in the gastrointestinal tract ALLERGAN, INC. (US) 1993-04-20 US disclosed
WO-1992013855-A1 (2-IMIDAZOLIN-2-YLAMINO) TETRAHYDROQUINOLAXINES AND METHODS FOR USING SAME ALLERGAN, INC. (US) 1992-08-20 WO disclosed
US-5089025-A HAIR DYE COMPOSITIONS AND CERTAIN 1,2,3,4-TETRAHYDRONITROQUINOXALINES USEFUL THEREIN HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1992-02-18 US disclosed
US-5077292-A Gastrointestinal disordes; kidney and vision defects ALLERGAN, INC. (US) 1991-12-31 US disclosed
US-5021416-A Glaucoma ALLERGAN, INC. (US) 1991-06-04 US disclosed
EP-0426719-A1 A HAIR DYE Henkel Kommanditgesellschaft auf Aktien (DE) 1991-05-15 EP disclosed
EP-0426390-A2 Method for using (2-imidazolin-2-ylamino) quinoxalines to reduce or maintain intraocular pressure ALLERGAN, INC. (US) 1991-05-08 EP disclosed
EP-0422878-A1 (2-Imidazolin-2-ylamino) tetrahydroquinoxalines and methods for using same ALLERGAN, INC. (US) 1991-04-17 EP disclosed
WO-1990001050-A1 A HAIR DYE HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1990-02-08 WO disclosed
EP-0353531-A1 Hair dye Henkel Kommanditgesellschaft auf Aktien (DE) 1990-02-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11180471-B2 Substituted oxopyridine derivatives OGFOD1, VASP, PNPO SMN1; SMN2 2641/4885HTT 1354/4885ALDH1A1 2345/4885
US-20250282748-A1 SUBSTITUTED OXOPYRIDINE DERIVATIVES OGFOD1, VASP, PNPO SMN1; SMN2 2641/4885HTT 1354/4885ALDH1A1 2345/4885
US-20230024752-A1 SUBSTITUTED OXOPYRIDINE DERIVATIVES OGFOD1, VASP, PNPO SMN1; SMN2 2641/4885HTT 1354/4885ALDH1A1 2345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.