SCHEMBL15519667

SCHEMBL15519667

CN1C(=O)C(C)(C)Oc2ccc(C(C)(c3ccc(-c4ccc(C(=O)O)c(F)c4)cc3Cl)C(O)C(F)(F)F)cc21

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12164169 0.80 PDE3B (0.34) PDE3BPDE3A
SCHEMBL474031 0.80 PDE3B (0.34) PDE3BPDE3A
SCHEMBL15520366 0.71 CYP11B2 (0.44)
SCHEMBL15520030 0.70 PDE3B (0.33) PDE3BPDE3A
SCHEMBL2816563 0.65 GPR55 (0.39) PDE3BPDE3A
SCHEMBL2817590 0.65 GPR55 (0.39) PDE3BPDE3A
SCHEMBL474393 0.65 GPR55 (0.39) PDE3BPDE3A
SCHEMBL12187874 0.65 NR1H2 (0.30)
SCHEMBL12164173 0.61 CPT2 (0.36)
SCHEMBL474367 0.61 CPT2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed