SCHEMBL15520282

SCHEMBL15520282

COC(=O)Oc1ccc(-c2ccc(C(C)C(O)(c3ccc4oc(=O)n(C)c4c3)C(F)(F)F)c(Cl)c2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 3/20 0.37
CTSC P53634 1/20 0.33
CYP11B2 P19099 1/20 0.33
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
KMO O15229 1/20 0.32
TP53 P04637 2/20 0.31
CUL4A Q13619 1/20 0.31
KCNJ1 P48048 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520208 0.95 GPR55 (0.36) GPR55CYP11B2POLBMAPTKMO
SCHEMBL15520636 0.94 GPR55 (0.35) GPR55CTSCCYP11B2MAPTKMO
SCHEMBL15520807 0.94 GPR55 (0.35) GPR55CTSCCYP11B2MAPTKMO
SCHEMBL15520263 0.94 GPR55 (0.35) GPR55CTSCCYP11B2MAPTKMO
SCHEMBL15520087 0.93 GPR55 (0.35) GPR55CYP11B2POLBMAPTKMO
SCHEMBL15520810 0.90 GPR55 (0.35) GPR55CTSCCYP11B2KMO
SCHEMBL12164093 0.90 GPR55 (0.37) GPR55CTSCCYP11B2KMOKCNJ1
SCHEMBL473982 0.90 GPR55 (0.37) GPR55CTSCCYP11B2KMOKCNJ1
SCHEMBL15520009 0.89 GPR55 (0.35) GPR55CYP11B2POLBKMO
SCHEMBL15520249 0.88 ALDH1A1 (0.35) GPR55CTSCCYP11B2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed