SCHEMBL15520249

SCHEMBL15520249

CCOC(=O)Oc1cc(-c2ccc(C(C)C(O)(c3ccc4oc(=O)n(C)c4c3)C(F)(F)F)c(Cl)c2)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TP53 P04637 2/20 0.35
GPR55 Q9Y2T6 3/20 0.35
CUL4A Q13619 1/20 0.33
POLB P06746 1/20 0.32
BDKRB1 P46663 3/20 0.31
KMO O15229 1/20 0.31
CYP11B2 P19099 1/20 0.31
CTSC P53634 1/20 0.30
EGFR P00533 1/20 0.30
KCNJ1 P48048 1/20 0.30
MAPT P10636 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520731 0.91 GPR55 (0.35) ALDH1A1TP53GPR55KMOCYP11B2
SCHEMBL15520282 0.88 GPR55 (0.37) TP53GPR55CUL4APOLBKMO
SCHEMBL12342539 0.88 ALDH1A1 (0.36) ALDH1A1TP53GPR55POLBBDKRB1
SCHEMBL12164097 0.88 ALDH1A1 (0.36) ALDH1A1TP53GPR55POLBBDKRB1
SCHEMBL473850 0.88 ALDH1A1 (0.36) ALDH1A1TP53GPR55POLBBDKRB1
SCHEMBL15520208 0.87 GPR55 (0.36) TP53GPR55CUL4APOLBKMO
SCHEMBL15520087 0.86 GPR55 (0.35) TP53GPR55POLBKMOCYP11B2
SCHEMBL15520708 0.85 CYP11B2 (0.38) ALDH1A1TP53GPR55POLBKMO
SCHEMBL15520636 0.85 GPR55 (0.35) GPR55KMOCYP11B2CTSCKCNJ1
SCHEMBL15520263 0.85 GPR55 (0.35) GPR55KMOCYP11B2CTSCKCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed