SCHEMBL15520702

SCHEMBL15520702

CCN1C(=O)COc2ccc(C(O)(C(C)c3ccc(-c4ccc(OC(=O)O)c(F)c4)cc3Cl)C(F)(F)F)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
HTT P42858 2/20 0.39
USP2 O75604 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
SLC5A1 P13866 3/20 0.37
SLC5A2 P31639 3/20 0.37
BRD4 O60885 1/20 0.36
POLB P06746 1/20 0.36
THRB P10828 1/20 0.35
KMO O15229 2/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
RORC P51449 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
OPRK1 P41145 1/20 0.33
UTS2R Q9UKP6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520272 0.95 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL15520261 0.95 USP2 (0.40) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL15520689 0.93 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL15520803 0.91 GPR55 (0.38) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL15520533 0.91 GPR55 (0.38) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL15520752 0.91 GPR55 (0.38) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL474334 0.90 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL12163929 0.90 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL474540 0.89 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR
SCHEMBL12163951 0.89 ALDH1A1 (0.41) ALDH1A1HTTUSP2L3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed