SCHEMBL15520261

SCHEMBL15520261

CCN1C(=O)COc2ccc(C(O)(C(C)c3ccc(-c4ccc(F)c(OC(=O)O)c4)cc3Cl)C(F)(F)F)cc21

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SLC5A1 P13866 3/20 0.38
SLC5A2 P31639 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
THRB P10828 1/20 0.36
KMO O15229 3/20 0.36
BRD4 O60885 1/20 0.36
POLB P06746 1/20 0.35
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520702 0.95 ALDH1A1 (0.40) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL15520689 0.94 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL15520272 0.93 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL15520532 0.91 GPR55 (0.38) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL12163951 0.89 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL474540 0.89 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL474334 0.88 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL12163929 0.88 ALDH1A1 (0.41) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL2815636 0.87 HTT (0.43) USP2HTTALDH1A1TSHRNPSR1
SCHEMBL474545 0.87 ALDH1A1 (0.42) USP2HTTALDH1A1TSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed