SCHEMBL15528720

SCHEMBL15528720

Cn1c(NC(=O)c2ccccc2)nnc1SCC(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.63
THRB P10828 1/20 0.57
TP53 P04637 2/20 0.56
GAA P10253 1/20 0.56
ALDH1A1 P00352 4/20 0.55
MAPT P10636 3/20 0.55
SENP1 Q9P0U3 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.54
PKM P14618 1/20 0.54
HTT P42858 2/20 0.54
MAPK1 P28482 2/20 0.54
RAB9A P51151 1/20 0.54
IDO1 P14902 1/20 0.53
HPGD P15428 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.53
KMT2A Q03164 1/20 0.52
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15528877 0.87 TDP1 (0.80) TDP1THRBTP53GAAALDH1A1
SCHEMBL4206372 0.80 PKM (0.85) ALDH1A1MAPTPKMHTTRAB9A
SCHEMBL4204258 0.77 MAPK1 (0.79) TDP1THRBTP53GAAALDH1A1
SCHEMBL3903365 0.77 GAA (0.76) TDP1THRBTP53GAAALDH1A1
SCHEMBL4207394 0.76 MAPK1 (0.64) TDP1THRBTP53GAAALDH1A1
SCHEMBL4208108 0.74 GAA (0.79) TDP1THRBTP53GAAMAPT
SCHEMBL4202666 0.74 GAA (0.86) TDP1GAAALDH1A1MAPK1NPSR1
SCHEMBL18559112 0.73 RECQL (0.81) TDP1THRBTP53GAAALDH1A1
SCHEMBL4216623 0.72 ALDH1A1 (0.72) TDP1ALDH1A1MAPTNPSR1KMT2A
SCHEMBL25132313 0.71 GAA (0.70) GAAALDH1A1MAPTSMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2850068-A1 GPR17 RECEPTOR MODULATORS. Universita' degli Studi di Milano (IT) 2015-03-25 EP disclosed
WO-2013167177-A1 GPR17 RECEPTOR MODULATORS. UNIVERSITA' DEGLI STUDI DI MILANO (IT) 2013-11-14 WO disclosed