SCHEMBL15529280

SCHEMBL15529280

CCOc1ccc(NC(=O)c2ccncc2NCc2ccccc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 4/20 0.58
KDM4E B2RXH2 4/20 0.58
KDM6B O15054 1/20 0.58
KDM4A O75164 1/20 0.58
KDM4D Q6B0I6 1/20 0.58
KMT2A Q03164 3/20 0.54
RAB9A P51151 9/20 0.54
NPC1 O15118 7/20 0.54
SMN1; SMN2 Q16637 5/20 0.54
TP53 P04637 5/20 0.54
POLB P06746 1/20 0.54
ALDH1A1 P00352 1/20 0.54
GAA P10253 1/20 0.54
ALOX15 P16050 1/20 0.54
LMNA P02545 2/20 0.53
PKM P14618 2/20 0.53
MEN1 O00255 2/20 0.53
HTT P42858 1/20 0.53
MITF O75030 1/20 0.53
NAMPT P43490 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15528663 0.92 KMT2A (0.54) KDM4EKMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL16625615 0.85 KDM4C (0.64) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL15529694 0.81 KDR (0.72) KDM4EKMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL18979244 0.77 KMT2A (0.64) KDM4EKMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL2087718 0.77 KDM4C (0.69) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL15528787 0.77 KMT2A (0.64) KDM4EKMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL16625601 0.77 ALDH1A1 (0.59) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL429479 0.76 KDR (0.66) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL4981514 0.76 KDR (0.74) KDM4CSMN1; SMN2POLBLMNAHTT
SCHEMBL4980164 0.76 NPC1 (0.66) KDM4EKMT2ARAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2846803-B1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF ALPHARMAGEN LLC (US) 2017-06-21 EP claimed
US-20150099758-A1 Alpha 7 Nicotinic Acetylcholine Receptor Allosteric Modulators, Their Derivatives and Uses Thereof ANVYL LLC (US) 2015-04-09 US claimed
EP-2846803-A1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF Anvyl, LLC (US) 2015-03-18 EP claimed
WO-2013169889-A1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF ANVYL LLC (US) 2013-11-14 WO claimed
EP-2846803-B1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF ALPHARMAGEN LLC (US) 2017-06-21 EP disclosed
EP-2846803-B1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF ALPHARMAGEN LLC (US) 2017-06-21 EP disclosed
US-20150099758-A1 Alpha 7 Nicotinic Acetylcholine Receptor Allosteric Modulators, Their Derivatives and Uses Thereof ANVYL LLC (US) 2015-04-09 US disclosed
US-20150099758-A1 Alpha 7 Nicotinic Acetylcholine Receptor Allosteric Modulators, Their Derivatives and Uses Thereof ANVYL LLC (US) 2015-04-09 US disclosed
EP-2846803-A1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF Anvyl, LLC (US) 2015-03-18 EP disclosed
WO-2013169889-A1 ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR ALLOSTERIC MODULATORS, THEIR DERIVATIVES AND USES THEREOF ANVYL LLC (US) 2013-11-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150099758-A1 Alpha 7 Nicotinic Acetylcholine Receptor Allosteric Modulators, Their Derivatives and Uses Thereof CHRNA7, CHRNA1, CHRNA2 KDM4C 3149/4885KDM4E 3133/4885KDM6B 2334/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.