SCHEMBL1552965

SCHEMBL1552965

COc1ccc(-n2c(CNC(=O)c3ccc(C(=O)O)cc3)nc3ccccc3c2=O)cc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.62
HTR7 P34969 5/20 0.61
ALDH1A1 P00352 1/20 0.61
MEN1 O00255 1/20 0.61
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
KMT2A Q03164 1/20 0.61
GAA P10253 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.56
MAPK1 P28482 1/20 0.55
PTGS2 P35354 1/20 0.54
UBE2N P61088 1/20 0.53
PTGER4 P35408 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL449634 0.97 ALDH1A1 (0.64) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL451191 0.95 ALDH1A1 (0.64) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL449655 0.93 POLB (0.61) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL447996 0.92 HTR7 (0.59) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL452387 0.91 HTR7 (0.59) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL450020 0.88 HTR7 (0.61) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL449587 0.85 SMN1; SMN2 (0.60) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL453594 0.82 ALDH1A1 (0.76) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL452084 0.81 PDE10A (0.60) PDE10AHTR7ALDH1A1MEN1CYP1A2
SCHEMBL450538 0.81 ALDH1A1 (0.66) PDE10AHTR7ALDH1A1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1521746-B1 QUINAZOLINONE MODULATORS OF NUCLEAR RECEPTORS X CEPTOR THERAPEUTICS INC (US) 2011-04-27 EP disclosed