SCHEMBL1553046

SCHEMBL1553046

CCOC(=O)c1sc(Cl)nc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
CYP1A2 P05177 1/20 0.54
HPGD P15428 5/20 0.50
TSHR P16473 1/20 0.50
MAPT P10636 4/20 0.45
TRPM8 Q7Z2W7 3/20 0.45
CDC7 O00311 2/20 0.43
DBF4 Q9UBU7 2/20 0.43
LMNA P02545 1/20 0.43
HSD17B10 Q99714 3/20 0.43
KDM4E B2RXH2 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
DHODH Q02127 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1505552 0.90 ALDH1A1 (0.66) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL1553063 0.87 ALDH1A1 (0.54) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL2826240 0.86 ALDH1A1 (0.53) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL9199229 0.83 ALDH1A1 (0.57) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL1553583 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL1554058 0.82 ALDH1A1 (0.49) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL27788399 0.81 ALDH1A1 (0.50) ALDH1A1HPGDTSHRMAPTTRPM8
SCHEMBL187316 0.81 ALDH1A1 (0.59) ALDH1A1HPGDTSHRMAPTCDC7
SCHEMBL28049117 0.81 ALDH1A1 (0.50) ALDH1A1CYP1A2HPGDTSHRMAPT
SCHEMBL1553145 0.81 SMN1; SMN2 (0.48) ALDH1A1CYP1A2HPGDTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735426-A1 HETEROAROMATIC DHODH INHIBITORS Immunic AG (DE) 2026-05-06 EP disclosed
WO-2025003402-A1 HETEROAROMATIC DHODH INHIBITORS IMMUNIC AG (DE) 2025-01-02 WO disclosed
EP-1853586-B1 ANTIBACTERIAL PIPERIDINE DERIVATIVES ASTRAZENECA AB (SE) 2013-07-24 EP disclosed
US-20130150366-A1 CHEMICAL COMPOUNDS ASTRAZENECA, INTELLECTUAL PROPERTY (GB) 2013-06-13 US disclosed
US-8399489-B2 Antibacterial piperdine derivatives ASTRAZENECA AB (GB) 2013-03-19 US disclosed
CN-101163693-B Antibacterial piperidine derivatives ASTRAZENECA AB 2013-03-06 CN disclosed
CN-102648199-A Piperidine compound and use thereof ASTRAZENECA AB 2012-08-22 CN disclosed
EP-2102199-B1 ANTIBACTERIAL POLYCYCLIC UREA COMPOUNDS ASTRAZENECA AB (SE) 2011-04-27 EP disclosed
EP-2102199-B1 ANTIBACTERIAL POLYCYCLIC UREA COMPOUNDS ASTRAZENECA AB (SE) 2011-04-27 EP disclosed
EP-2158199-B1 PIPERIDINE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2010-11-17 EP disclosed
WO-2008152418-A1 PIPERIDINE COMPOUNDS AND USES THEREOF ASTRAZENECA AB (SE) 2008-12-18 WO disclosed
WO-2008068470-A1 ANTIBACTERIAL POLYCYCLIC UREA COMPOUNDS ASTRAZENECA AB (SE) 2008-06-12 WO disclosed
WO-2008068470-A1 ANTIBACTERIAL POLYCYCLIC UREA COMPOUNDS ASTRAZENECA AB (SE) 2008-06-12 WO disclosed
US-20080132546-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2008-06-05 US disclosed
US-20080132546-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2008-06-05 US disclosed
US-20080132546-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2008-06-05 US disclosed
CN-101163693-A Antibacterial piperidine derivatives ASTRAZENECA AB (SE) 2008-04-16 CN disclosed
WO-2008020222-A1 PYRROLE DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2008-02-21 WO disclosed
EP-1853586-A1 ANTIBACTERIAL PIPERIDINE DERIVATIVES AstraZeneca AB (SE) 2007-11-14 EP disclosed
WO-2006087543-A1 ANTIBACTERIAL PIPERIDINE DERIVATIVES ASTRAZENECA AB (SE) 2006-08-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130150366-A1 CHEMICAL COMPOUNDS MRPL21, NISCH, CFTR ALDH1A1 419/4885CYP1A2 33/4885HPGD 429/4885
US-20080132546-A1 CHEMICAL COMPOUNDS MRPL21, NISCH, ABCB11 ALDH1A1 488/4885CYP1A2 41/4885HPGD 389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.