SCHEMBL15533812

SCHEMBL15533812

COc1ccc(-c2cc(Nc3c(F)c(F)c(F)c(F)c3F)ncn2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP1A2 P05177 4/20 0.46
CYP2D6 P10635 4/20 0.46
CYP2C19 P33261 4/20 0.46
CLK4 Q9HAZ1 4/20 0.46
HSD17B10 Q99714 3/20 0.46
LMNA P02545 3/20 0.46
USP2 O75604 2/20 0.46
ALOX15 P16050 2/20 0.46
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
RAB9A P51151 4/20 0.43
TSHR P16473 3/20 0.43
TP53 P04637 2/20 0.43
MAPK1 P28482 2/20 0.43
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
TNF P01375 1/20 0.43
HTT P42858 1/20 0.43
CCR6 P51684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10685065 0.83 MEN1 (0.46) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533528 0.79 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533525 0.78 MEN1 (0.62) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533795 0.78 ABL1 (0.64) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15534515 0.77 MAPT (0.44) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533950 0.77 ABL1 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533672 0.76 MAPT (0.48) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL5923911 0.76 TRPV1 (0.56) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15533631 0.76 ABL1 (0.46) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4
SCHEMBL15534052 0.76 EGFR (0.55) ALDH1A1CYP1A2CYP2D6CYP2C19CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO claimed
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed