Bergapten

Bergapten

SCHEMBL15534211

COc1c2ccoc2cc2oc(=O)ccc12.COc1cc2occc2c2oc(=O)ccc12

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.82
CYP3A4 P08684 6/20 0.82
KDM4E B2RXH2 5/20 0.82
MAPT P10636 2/20 0.82
CYP1B1 Q16678 3/20 0.78
CYP1A1 P04798 2/20 0.78
CYP1A2 P05177 2/20 0.78
CYP2A6 P11509 2/20 0.78
HSD17B10 Q99714 2/20 0.78
PGR P06401 1/20 0.78
ADORA3 P0DMS8 1/20 0.78
CYP2D6 P10635 1/20 0.78
CYP2C9 P11712 1/20 0.78
KCNA2 P16389 1/20 0.78
TSHR P16473 1/20 0.78
MAOA P21397 1/20 0.78
CYP2C19 P33261 1/20 0.78
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isobergaptene SCHEMBL2253427 0.91 CYP3A4 (1.00) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
Bergapten SCHEMBL4731782 0.88 ALDH1A1 (1.00) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
Bergapten SCHEMBL50066 0.88 ALDH1A1 (1.00) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
Bergapten SCHEMBL29529284 0.88 ALDH1A1 (1.00) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
Isopimpinellin SCHEMBL29787210 0.85 CYP3A4 (0.82) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
Bergapten SCHEMBL9792363 0.81 CYP3A4 (0.74) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
5,6,7-Trimethoxycoumarin SCHEMBL4743900 0.76 ALDH1A1 (0.62) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
SCHEMBL19346062 0.74 ALDH1A1 (0.72) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
SCHEMBL5794191 0.73 CA12 (1.00) ALDH1A1CYP3A4KDM4EMAPTCYP1B1
SCHEMBL9122678 0.73 ALDH1A1 (0.71) ALDH1A1CYP3A4KDM4ECYP1B1CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013176955-A1 CARDIOPROTECTIVE COMPOUNDS, THEIR USE WITH CHEMOTHERAPY, AND METHODS FOR IDENTIFYING THEM THE GENERAL HOSPITAL CORPORATION (US) 2013-11-28 WO disclosed