SCHEMBL15535856

SCHEMBL15535856

COc1c(NC(C)=O)cccc1B(O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
IDO1 P14902 1/20 0.45
TSHR P16473 1/20 0.45
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAOA P21397 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
POLB P06746 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTK2 Q05397 1/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CASR P41180 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14046286 0.83 ALDH1A1 (0.61) KDM4ECYP1A2CYP2C9IDO1TSHR
SCHEMBL6774791 0.79 BRD4 (0.55) KDM4ECYP1A2CYP2C9IDO1TSHR
SCHEMBL29469169 0.78 ALDH1A1 (0.59) KDM4ECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL521100 0.78 ALDH1A1 (0.59) KDM4ECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL8374069 0.78 KDM4E (0.46) KDM4ECYP1A2CYP2C9IDO1TSHR
SCHEMBL2549708 0.77 ALDH1A1 (0.53) KDM4ETSHRALDH1A1HPGDSMN1; SMN2
SCHEMBL3792891 0.77 ALDH1A1 (0.48) KDM4ECYP1A2TSHRALDH1A1HPGD
SCHEMBL22587415 0.77 ALDH1A1 (0.48) KDM4ETSHRALDH1A1HPGDSMN1; SMN2
SCHEMBL13255390 0.77 LMNA (0.51) KDM4ECYP1A2CYP2C9IDO1TSHR
SCHEMBL3585917 0.76 ALDH1A1 (0.47) KDM4ETSHRALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855483-A1 PYRROLOPYRROLIDINONE COMPOUNDS Novartis AG (CH) 2015-04-08 EP disclosed
WO-2013175417-A1 PYRROLOPYRROLIDINONE COMPOUNDS NOVARTIS AG (CH) 2013-11-28 WO disclosed