SCHEMBL15536378

SCHEMBL15536378

COc1ccc(COCC2=CCCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.51
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
GAA P10253 1/20 0.47
KMT2A Q03164 3/20 0.45
TSHR P16473 2/20 0.45
MEN1 O00255 2/20 0.45
IDO1 P14902 2/20 0.44
AGXT P21549 2/20 0.44
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
APP P05067 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9414387 0.80 ALDH1A1 (0.40) ALDH1A1RAB9ASMN1; SMN2
SCHEMBL10881311 0.78 CXCR3 (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL10881315 0.78 CXCR3 (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL10881322 0.78 CXCR3 (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL34413 0.78 IDO1 (0.67) ALDH1A1SMN1; SMN2TSHRIDO1AGXT
Methoxymethane SCHEMBL28823290 0.76 IDO1 (0.64) ALDH1A1SMN1; SMN2TSHRIDO1AGXT
Bromide SCHEMBL28558295 0.76 IDO1 (0.64) ALDH1A1SMN1; SMN2TSHRIDO1AGXT
Hydrochloric Acid SCHEMBL28912134 0.76 IDO1 (0.68) ALDH1A1SMN1; SMN2TSHRIDO1AGXT
Potassium SCHEMBL1477050 0.76 IDO1 (0.64) ALDH1A1SMN1; SMN2TSHRIDO1AGXT
SCHEMBL1475481 0.76 IDO1 (0.64) ALDH1A1SMN1; SMN2TSHRIDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855428-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN Genentech, Inc. (US) 2015-04-08 EP disclosed
US-8952169-B2 N-substituted benzamides and methods of use thereof XENON PHARMACEUTICALS INC. (CA) 2015-02-10 US disclosed
US-8952169-B2 N-substituted benzamides and methods of use thereof XENON PHARMACEUTICALS INC. (CA) 2015-02-10 US disclosed
WO-2013177224-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN GENENTECH, INC. (US) 2013-11-28 WO disclosed