SCHEMBL15536619

SCHEMBL15536619

COc1ccc(COCC2CC=CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.47
AGXT P21549 2/20 0.47
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
TRPV6 Q9H1D0 1/20 0.43
APP P05067 7/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAOB P27338 1/20 0.41
CALM1 P0DP23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22288217 0.80 L3MBTL1 (0.54) IDO1AGXTCA1CA2APP
SCHEMBL16686216 0.79 IDO1 (0.43) IDO1AGXTCA1CA2TRPV6
SCHEMBL880157 0.78 TSHR (0.54)
SCHEMBL34413 0.77 IDO1 (0.67) IDO1AGXTCA1CA2APP
SCHEMBL16685703 0.76 IDO1 (0.41) IDO1AGXTCA1CA2TRPV6
SCHEMBL16448677 0.76 IDO1 (0.41) IDO1AGXTCA1CA2TRPV6
SCHEMBL3049370 0.76 NAAA (0.43) IDO1AGXTCA1CA2TRPV6
SCHEMBL16448678 0.76 IDO1 (0.41) IDO1AGXTCA1CA2TRPV6
Methyl Alcohol SCHEMBL8601404 0.76 CA1 (0.42) IDO1AGXTCA1CA2TRPV6
SCHEMBL15794308 0.76 IDO1 (0.47) IDO1AGXTCA1CA2TRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855428-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN Genentech, Inc. (US) 2015-04-08 EP disclosed
US-8952169-B2 N-substituted benzamides and methods of use thereof XENON PHARMACEUTICALS INC. (CA) 2015-02-10 US disclosed
US-8952169-B2 N-substituted benzamides and methods of use thereof XENON PHARMACEUTICALS INC. (CA) 2015-02-10 US disclosed
WO-2013177224-A1 N-SUBSTITUTED BENZAMIDES AND THEIR USE IN THE TREATMENT OF PAIN GENENTECH, INC. (US) 2013-11-28 WO disclosed