SCHEMBL15538366

SCHEMBL15538366

CC(C)(C)N1CCC(COc2ccc(-c3ccc(S(C)(=O)=O)cc3)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.49
GPR183 P32249 1/20 0.46
PTGS2 P35354 4/20 0.45
PTGS1 P23219 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15539741 0.86 KCNH2 (0.43) GPR119GPR183PTGS2PTGS1
SCHEMBL15538238 0.83 GPR119 (0.48) GPR119GPR183
SCHEMBL15538188 0.83 GPR119 (0.46) GPR119GPR183PTGS2PTGS1
SCHEMBL15538548 0.83 GPR119 (0.46) GPR119GPR183PTGS2PTGS1
SCHEMBL21534611 0.82 PTGS2 (0.47) GPR119GPR183PTGS2PTGS1
SCHEMBL15539139 0.82 PTGS2 (0.46) GPR119GPR183PTGS2PTGS1
SCHEMBL389015 0.82 GPR119 (0.75) GPR119
SCHEMBL16803722 0.81 GPR119 (0.48) GPR119GPR183
SCHEMBL388606 0.81 GPR119 (0.46) GPR119GPR183PTGS2PTGS1
SCHEMBL13589518 0.81 PTGS2 (0.53) GPR119PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2858986-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST Chong Kun Dang Pharmaceutical Corp. (KR) 2015-04-15 EP disclosed
WO-2013187646-A1 PIPERIDINE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2013-12-19 WO disclosed