SCHEMBL15544285

SCHEMBL15544285

O=C1COC2(CCN(Cc3ccc(-c4ccc5cnccc5c4)cc3F)CC2)CN1C1CC1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FASN P49327 11/20 0.65
OPRM1 P35372 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD11B1 P28845 1/20 0.34
CYP2D6 P10635 1/20 0.33
GPR6 P46095 1/20 0.33
PDE2A O00408 2/20 0.33
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543510 0.97 FASN (0.60) FASNOPRM1SIGMAR1ALDH1A1MAPK1
SCHEMBL15581938 0.89 FASN (0.49) FASNOPRM1SIGMAR1ALDH1A1CHRM1
SCHEMBL15543306 0.89 FASN (0.49) FASNOPRM1SIGMAR1ALDH1A1
SCHEMBL15544827 0.87 FASN (0.49) FASNOPRM1SIGMAR1ALDH1A1MAPK1
SCHEMBL15543784 0.87 FASN (0.50) FASNOPRM1SIGMAR1ALDH1A1MAPK1
SCHEMBL15544087 0.84 FASN (0.48) FASNOPRM1SIGMAR1ALDH1A1CHRM1
SCHEMBL14842076 0.84 FASN (0.65) FASNOPRM1SIGMAR1HSD11B1CHRM1
SCHEMBL15543780 0.84 FASN (0.51) FASNOPRM1SIGMAR1ALDH1A1MAPK1
SCHEMBL15543468 0.84 FASN (0.57) FASNOPRM1SIGMAR1CHRM1
SCHEMBL15544977 0.84 FASN (0.51) FASNOPRM1SIGMAR1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO claimed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed