SCHEMBL15544827

SCHEMBL15544827

O=C1COC2(CCN(Cc3ccc(-c4ccc5ncncc5c4)cc3F)CC2)CN1C1CC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FASN P49327 6/20 0.49
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HSD11B1 P28845 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
PDE4A P27815 1/20 0.33
OPRM1 P35372 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
BTK Q06187 1/20 0.32
PDE2A O00408 2/20 0.32
ACVRL1 P37023 2/20 0.32
ACVR1 Q04771 2/20 0.32
BMPR1A P36894 1/20 0.32
CHRM1 P11229 3/20 0.32
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543784 0.94 FASN (0.50) FASNCYP1A2CYP3A4HSD11B1ALDH1A1
SCHEMBL15543468 0.88 FASN (0.57) FASNOPRM1SIGMAR1CHRM1
SCHEMBL15543510 0.87 FASN (0.60) FASNHSD11B1ALDH1A1MAPK1OPRM1
SCHEMBL15544285 0.87 FASN (0.65) FASNHSD11B1ALDH1A1MAPK1OPRM1
SCHEMBL15544977 0.86 FASN (0.51) FASNHSD11B1ALDH1A1MAPK1OPRM1
SCHEMBL15543780 0.85 FASN (0.51) FASNHSD11B1ALDH1A1MAPK1OPRM1
SCHEMBL15581938 0.84 FASN (0.49) FASNALDH1A1OPRM1SIGMAR1CHRM1
SCHEMBL15543306 0.84 FASN (0.49) FASNALDH1A1OPRM1SIGMAR1
SCHEMBL15543479 0.83 FASN (0.48) FASNHSD11B1ALDH1A1MAPK1OPRM1
SCHEMBL15543457 0.83 FASN (0.49) FASNHSD11B1ALDH1A1MAPK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO claimed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed