SCHEMBL15544928

SCHEMBL15544928

Cc1cc([N+](=O)[O-])cnc1N(C)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
GAA P10253 4/20 0.42
HTT P42858 3/20 0.42
TDP1 Q9NUW8 3/20 0.39
TSHR P16473 1/20 0.39
ATM Q13315 1/20 0.38
GPR35 Q9HC97 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15544924 1.00 ALDH1A1 (0.48) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL15545142 0.92 ALDH1A1 (0.42) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL15545143 0.92 ALDH1A1 (0.42) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL9112475 0.86 ALDH1A1 (0.46) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL9112479 0.86 ALDH1A1 (0.46) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL1100036 0.82 ALDH1A1 (0.62) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL15545493 0.81 ALDH1A1 (0.45) ALDH1A1HTTMAPTKMT2A
SCHEMBL1163006 0.81 ALDH1A1 (0.45) ALDH1A1GAAHTTTDP1TSHR
SCHEMBL15545495 0.81 ALDH1A1 (0.45) ALDH1A1HTTMAPTKMT2A
SCHEMBL16679829 0.81 ALDH1A1 (0.45) ALDH1A1GAAHTTGPR35CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870144-A1 OREXIN RECEPTOR ANTAGONISTS Heptares Therapeutics Limited (GB) 2015-05-13 EP disclosed
WO-2014006402-A1 OREXIN RECEPTOR ANTAGONISTS HEPTARES THERAPEUTICS LIMITED (GB) 2014-01-09 WO disclosed