SCHEMBL15545495

SCHEMBL15545495

COc1cc([N+](=O)[O-])cnc1N(C)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HTT P42858 3/20 0.44
PKM P14618 3/20 0.44
KMT2A Q03164 7/20 0.42
MEN1 O00255 3/20 0.42
MAPT P10636 3/20 0.42
GLA P06280 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 2/20 0.40
ERN1 O75460 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545493 1.00 ALDH1A1 (0.45) ALDH1A1HTTPKMKMT2AMEN1
SCHEMBL16680759 0.83 ALDH1A1 (0.43) ALDH1A1HTTPKMKMT2AMEN1
SCHEMBL15544924 0.81 ALDH1A1 (0.48) ALDH1A1HTTKMT2AMAPT
SCHEMBL15544928 0.81 ALDH1A1 (0.48) ALDH1A1HTTKMT2AMAPT
SCHEMBL15545353 0.78 ALDH1A1 (0.39) ALDH1A1HTTPKMKMT2AMEN1
SCHEMBL15544895 0.77 ALDH1A1 (0.41) ALDH1A1HTTPKMKMT2AMEN1
SCHEMBL15545143 0.75 ALDH1A1 (0.42) ALDH1A1HTTKMT2AMEN1MAPT
SCHEMBL15545142 0.75 ALDH1A1 (0.42) ALDH1A1HTTKMT2AMEN1MAPT
SCHEMBL3648669 0.74 ERN1 (0.50) ALDH1A1HTTPKMKMT2AMEN1
SCHEMBL29865611 0.72 HTT (0.50) ALDH1A1HTTPKMKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870144-A1 OREXIN RECEPTOR ANTAGONISTS Heptares Therapeutics Limited (GB) 2015-05-13 EP disclosed
WO-2014006402-A1 OREXIN RECEPTOR ANTAGONISTS HEPTARES THERAPEUTICS LIMITED (GB) 2014-01-09 WO disclosed