SCHEMBL15545142

SCHEMBL15545142

Cc1cc([N+](=O)[O-])cnc1Cl.Cc1cc([N+](=O)[O-])cnc1N(C)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
GAA P10253 3/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 2/20 0.33
GPR35 Q9HC97 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
TSHR P16473 1/20 0.33
F2 P00734 1/20 0.33
PLAU P00749 1/20 0.33
KLKB1 P03952 1/20 0.33
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545143 1.00 ALDH1A1 (0.42) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL15544924 0.92 ALDH1A1 (0.48) ALDH1A1GAAHTTKMT2AMAPT
SCHEMBL15544928 0.92 ALDH1A1 (0.48) ALDH1A1GAAHTTKMT2AMAPT
SCHEMBL31143401 0.82 ALDH1A1 (0.47) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL801244 0.82 ALDH1A1 (0.47) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL26928548 0.80 ALDH1A1 (0.40) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL9112475 0.79 ALDH1A1 (0.46) ALDH1A1GAAHTTMAPTTDP1
SCHEMBL9112479 0.79 ALDH1A1 (0.46) ALDH1A1GAAHTTMAPTTDP1
SCHEMBL1100036 0.76 ALDH1A1 (0.62) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL15545495 0.75 ALDH1A1 (0.45) ALDH1A1HTTMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870144-A1 OREXIN RECEPTOR ANTAGONISTS Heptares Therapeutics Limited (GB) 2015-05-13 EP disclosed
WO-2014006402-A1 OREXIN RECEPTOR ANTAGONISTS HEPTARES THERAPEUTICS LIMITED (GB) 2014-01-09 WO disclosed