SCHEMBL15548752

SCHEMBL15548752

COc1ccc(CC(=O)O)c(Br)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
HSD17B10 Q99714 1/20 0.41
NNMT P40261 2/20 0.39
PTGS1 P23219 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
KDM4E B2RXH2 4/20 0.36
MTNR1A P48039 4/20 0.36
MTNR1B P49286 4/20 0.36
ALDH1A1 P00352 2/20 0.36
ABL1 P00519 1/20 0.36
MAPT P10636 1/20 0.36
RECQL P46063 1/20 0.36
RIN1 Q13671 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36
GAA P10253 2/20 0.35
MMP2 P08253 1/20 0.35
MMP8 P22894 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28699694 0.85 POLB (0.39) POLBTDP1HSD17B10NNMTKDM4E
SCHEMBL30034021 0.80 POLB (0.44) POLBTDP1HSD17B10NNMTPTGS1
SCHEMBL20565255 0.80 POLB (0.44) POLBTDP1HSD17B10NNMTPTGS1
SCHEMBL30486603 0.79 PDE4A (0.38) POLBTDP1NNMTKDM4EMTNR1A
SCHEMBL21383732 0.79 PDE4A (0.38) POLBTDP1NNMTKDM4EMTNR1A
SCHEMBL30564474 0.77 SRC (0.41) POLBTDP1HSD17B10PTGS1PTGDR2
SCHEMBL21383820 0.77 CYP1A2 (0.37) POLBTDP1NNMTMTNR1AMTNR1B
SCHEMBL30529295 0.77 CYP1A2 (0.37) POLBTDP1NNMTMTNR1AMTNR1B
SCHEMBL28045757 0.74 TDP1 (0.66) POLBTDP1HSD17B10NNMTKDM4E
SCHEMBL3149015 0.72 MTNR1A (0.41) POLBTDP1PTGS1AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2855483-A1 PYRROLOPYRROLIDINONE COMPOUNDS Novartis AG (CH) 2015-04-08 EP disclosed
WO-2013175417-A1 PYRROLOPYRROLIDINONE COMPOUNDS NOVARTIS AG (CH) 2013-11-28 WO disclosed