SCHEMBL28699694

SCHEMBL28699694

COC(=O)Cc1ccc(OC)nc1Br

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TXNRD1 Q16881 1/20 0.39
NNMT P40261 2/20 0.38
MTNR1A P48039 11/20 0.38
MTNR1B P49286 11/20 0.38
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 1/20 0.36
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15548752 0.85 POLB (0.44) POLBTDP1NNMTMTNR1AMTNR1B
SCHEMBL30486603 0.78 PDE4A (0.38) POLBTDP1TXNRD1NNMTMTNR1A
SCHEMBL21383732 0.78 PDE4A (0.38) POLBTDP1TXNRD1NNMTMTNR1A
SCHEMBL28594753 0.77 KDM4E (0.39) POLBTDP1TXNRD1NNMTMTNR1A
SCHEMBL30529295 0.75 CYP1A2 (0.37) POLBTDP1TXNRD1NNMTMTNR1A
SCHEMBL21383820 0.75 CYP1A2 (0.37) POLBTDP1TXNRD1NNMTMTNR1A
SCHEMBL25679572 0.75 CYP4F2 (0.38) POLBCYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL20487887 0.74 ALDH1A1 (0.40) CYP4F2CYP4A11KDM4EALDH1A1MAPT
SCHEMBL8998233 0.72 KDM4E (0.43) TDP1CYP4F2CYP4A11KDM4EALDH1A1
SCHEMBL14880583 0.72 MTNR1A (0.65) TXNRD1MTNR1AMTNR1BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118317951-A Phthalazine derivatives as pyruvate kinase modulators 西特瑞治疗有限公司 2024-07-09 CN disclosed
CN-113354635-B Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2023-04-18 CN disclosed
CN-113354635-A Pyrrolidine integrin regulator and application thereof 清药同创(北京)药物研发中心有限公司 2021-09-07 CN disclosed