SCHEMBL155647

SCHEMBL155647

CC1CCc2ccccc2O1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.44
HTR1A P08908 4/20 0.42
SIGMAR1 Q99720 2/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
CA1 P00915 1/20 0.40
CA9 Q16790 1/20 0.40
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
HTR1D P28221 2/20 0.39
SSTR4 P31391 1/20 0.39
HPGD P15428 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
PDPK1 O15530 1/20 0.37
NISCH Q9Y2I1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17167266 1.00 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL16429469 1.00 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL799675 1.00 CA2 (0.44) CA2HTR1ASIGMAR1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL27611840 0.98 CA2 (0.43) CA2HTR1ASIGMAR1ADRA2AADRA2B
Ammonia Solution, Strong SCHEMBL27679026 0.98 CA2 (0.43) CA2HTR1ASIGMAR1ADRA2AADRA2B
Ammonia Solution, Strong SCHEMBL27347848 0.98 CA2 (0.43) CA2HTR1ASIGMAR1ADRA2AADRA2B
Methyl Alcohol SCHEMBL20819455 0.96 CA2 (0.42) CA2HTR1ASIGMAR1ADRA2AADRA2B
Pyrimidine SCHEMBL27469036 0.87 HTR1A (0.41) CA2HTR1ASIGMAR1ADRA2AADRA2B
SCHEMBL18473078 0.85 PTGS2 (0.36) CA2CA1CA9BRD4CREBBP
SCHEMBL24926978 0.85 TSHR (0.41) CA2HTR1ASIGMAR1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 183 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100430391-C Method for producing 2-[-5-(4-fluoprophenyl)-3-pyridylmethylaminomethyl]-chromane MERCK PATENT GMBH (DE) 2008-11-05 CN claimed
CN-1246319-C Amino (thio) ether derivative MERCK PATENT AG (DE) 2006-03-22 CN claimed
CN-1622944-A Method for producing 2-[-5-(4-fluoprophenyl)-3-pyridylmethylaminomethyl]-chromane MERCK PATENT GMBH (DE) 2005-06-01 CN claimed
CN-1564818-A Stereoselective synthesis method of 2-hydroxymethyl-chroman WYETH CORP (US) 2005-01-12 CN claimed
CN-1561337-A Stereospecific process for the synthesis of 2-yl chroman derivatives WYETH CORP (US) 2005-01-05 CN claimed
CN-1451001-A Chromanone derivatives MERCK PATENT GMBH (DE) 2003-10-22 CN claimed
CN-1067389-C Benzodihydropyran assorbic acid derivatives, their preparation and use BASF AG (DE) 2001-06-20 CN claimed
WO-2000012082-A1 FORMAMIDE COMPOUNDS AS THERAPEUTIC AGENTS GLAXO GROUP LIMITED (GB) 2000-03-09 WO claimed
EP-0759750-A4 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1998-05-27 EP claimed
CN-1177596-A Benzodihydropyran assorbic acid derivatives, their preparation and use BASF AG (DE) 1998-04-01 CN claimed
EP-0759750-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO, Howard, K. (US) 1997-03-05 EP claimed
WO-1995031194-A1 COMPOSITIONS FOR TREATMENT OF CHRONIC INFLAMMATORY DISEASES SHAPIRO HOWARD K (US) 1995-11-23 WO claimed
WO-2024059951-A1 INHIBITORS OF THE ANDROGEN RECEPTOR DNA-BINDING DOMAIN THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2024-03-28 WO disclosed
CN-117377669-A TYK2 inhibitor and application thereof 苏多生物科学有限公司 2024-01-09 CN disclosed
EP-3826723-B1 BORONIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2023-10-18 EP disclosed
WO-2023091554-A1 NOVEL HETEROARYL-UREA COMPOUNDS AS KV7.2 INHIBITORS ICAGEN, LLC (US) 2023-05-25 WO disclosed
US-5703115-A VASOCONSTRICTORS JANSSEN PHARMACEUTICA, N.V. (BE) 1997-12-30 US disclosed
WO-1997047617-A1 ENANTIOMER SEPARATION FROM CHROMANE ACID ESTERS MERCK PATENT GMBH (DE) 1997-12-18 WO disclosed
US-5688952-A VASOCONSTRICTOR INTERMEDIATES JANSSEN PHARMACEUTICA, N.V. (BE) 1997-11-18 US disclosed
CN-1034416-Y With comfortable kinin antagonists for the preparation method of peptide He toru spa 1997-04-02 CN disclosed