SCHEMBL1556671

SCHEMBL1556671

O=C(C=Cc1cncs1)c1ccncc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 4/20 0.53
CYP1A1 P04798 9/20 0.47
CYP1A2 P05177 9/20 0.47
CYP2D6 P10635 9/20 0.47
CYP1B1 Q16678 9/20 0.47
HTT P42858 1/20 0.46
MAPT P10636 4/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
NPY1R P25929 1/20 0.46
MAPK1 P28482 1/20 0.46
NPY2R P49146 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.45
HDAC6 Q9UBN7 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PSMD14 O00487 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP2C8 P10632 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1555817 0.77 CYP1B1 (0.59) CYP1A1CYP1A2CYP2D6CYP1B1MAPT
SCHEMBL2522174 0.75 HCAR2 (0.48) SMN1; SMN2MAPK1HDAC6KMT2A
SCHEMBL2522171 0.75 HCAR2 (0.48) SMN1; SMN2MAPK1HDAC6KMT2A
SCHEMBL6997673 0.74 HTT (0.67) PFKFB3CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL6997670 0.74 HTT (0.67) PFKFB3CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL4572963 0.74 GLA (0.38) CYP1A2HTTMAPTSMN1; SMN2ALDH1A1
SCHEMBL18985284 0.74 CCNC (0.41) HTTMAPTSMN1; SMN2ALDH1A1MEN1
SCHEMBL4572964 0.74 GLA (0.38) CYP1A2HTTMAPTSMN1; SMN2ALDH1A1
SCHEMBL6934856 0.73 CYP1B1 (0.70) PFKFB3CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL6934854 0.73 CYP1B1 (0.70) PFKFB3CYP1A1CYP1A2CYP2D6CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488533-A1 IMIDAZOTHIAZOLE-CHALCONE DERIVATIVES AS POTENTIAL ANTICANCER AGENTS AND PROCESS FOR THE PREPARATION THEREOF Council of Scientific & Industrial Research (IN) 2012-08-22 EP claimed
WO-2011045646-A1 IMIDAZOTHIAZOLE-CHALCONE DERIVATIVES AS POTENTIAL ANTICANCER AGENTS AND PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2011-04-21 WO claimed