SCHEMBL6997670

SCHEMBL6997670

O=C(/C=C/C(=O)c1ccncc1)c1ccncc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.67
PFKFB3 Q16875 2/20 0.58
NAPRT Q6XQN6 1/20 0.56
CYP1A1 P04798 9/20 0.55
CYP1A2 P05177 9/20 0.55
CYP2D6 P10635 9/20 0.55
CYP1B1 Q16678 9/20 0.55
GPR52 Q9Y2T5 1/20 0.55
ALDH1A1 P00352 5/20 0.53
HPGD P15428 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MAPT P10636 1/20 0.53
NPY1R P25929 1/20 0.53
MAPK1 P28482 1/20 0.53
NPY2R P49146 1/20 0.53
PKM P14618 2/20 0.52
ATM Q13315 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997673 1.00 HTT (0.67) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL27687985 0.86 HTT (0.63) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL6934854 0.84 CYP1B1 (0.70) HTTPFKFB3CYP1A1CYP1A2CYP2D6
SCHEMBL6934856 0.84 CYP1B1 (0.70) HTTPFKFB3CYP1A1CYP1A2CYP2D6
SCHEMBL8501319 0.82 ALDH1A1 (0.58) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL2999914 0.81 ALDH1A1 (0.55) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL1863 0.81 HTT (1.00) HTTCYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL11007423 0.81 HTT (0.53) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL2999911 0.81 ALDH1A1 (0.55) HTTPFKFB3NAPRTCYP1A1CYP1A2
SCHEMBL11005951 0.81 HTT (0.53) HTTPFKFB3NAPRTCYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0921119-B1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2003-07-02 EP disclosed
US-6114360-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-09-05 US disclosed
US-6063804-A Pyrrole compounds ADIR ET COMPAGNIE (FR) 2000-05-16 US disclosed
EP-0921119-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1999-06-09 EP disclosed