SCHEMBL18985284

SCHEMBL18985284

NC(=O)C=Cc1cncs1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 2/20 0.41
CDK8 P49336 2/20 0.41
NLRP3 Q96P20 1/20 0.36
HCAR2 Q8TDS4 1/20 0.35
PIM1 P11309 1/20 0.35
RAB9A P51151 4/20 0.34
NPC1 O15118 3/20 0.34
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
CYP19A1 P11511 1/20 0.32
HDAC8 Q9BY41 1/20 0.31
MEN1 O00255 1/20 0.31
PSMD14 O00487 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
GLA P06280 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2522171 0.82 HCAR2 (0.48) NLRP3HCAR2PIM1RAB9ANPC1
SCHEMBL2522174 0.82 HCAR2 (0.48) NLRP3HCAR2PIM1RAB9ANPC1
SCHEMBL4395610 0.82
SCHEMBL4572963 0.81 GLA (0.38) NLRP3HCAR2PIM1RAB9ANPC1
SCHEMBL4572964 0.81 GLA (0.38) NLRP3HCAR2PIM1RAB9ANPC1
SCHEMBL9255626 0.77 KMT2A (0.49) CCNCCDK8NLRP3HCAR2RAB9A
SCHEMBL9255628 0.77 KMT2A (0.49) CCNCCDK8NLRP3HCAR2RAB9A
SCHEMBL6297811 0.77 PIK3CD (0.37) NLRP3PIM1RAB9ASMN1; SMN2CYP19A1
SCHEMBL1556671 0.74 PFKFB3 (0.53) SMN1; SMN2ALDH1A1MEN1PSMD14LMNA
SCHEMBL17926074 0.73 RAB9A (0.47) CCNCCDK8HCAR2RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017102014-A1 PROPENAMIDE THIOPHENE DERIVATIVES AS FLAVIVIRUS INHIBITORS AND THEIR USE UNIVERSITE D'AIX-MARSEILLE (FR) 2017-06-22 WO disclosed