SCHEMBL15568002

SCHEMBL15568002

CCN(CCCNC(=O)C1CCN(c2nc3ccccc3n2Cc2ccc(C)cc2)CC1)c1cccc(C)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2C19 P33261 1/20 0.60
GFER P55789 2/20 0.58
TP53 P04637 5/20 0.57
HTT P42858 1/20 0.57
ALDH1A1 P00352 2/20 0.56
KMT2A Q03164 3/20 0.52
HRH1 P35367 3/20 0.51
KCNH2 Q12809 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51
MAPT P10636 2/20 0.51
POLB P06746 1/20 0.51
ALOX15 P16050 1/20 0.51
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.48
HTR3A P46098 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15567362 0.76 HRH1 (0.69) CYP2D6HTTALDH1A1KMT2AHRH1
SCHEMBL15452490 0.73 HRH1 (0.65) CYP2D6CYP3A4ALDH1A1HRH1KCNH2
SCHEMBL18286772 0.73 CYP1A2 (0.71) CYP2D6CYP1A2CYP3A4CYP2C19GFER
Trifluoroacetic Acid SCHEMBL15568340 0.73 HRH1 (0.53) CYP2D6HRH1KCNH2HTR3A
SCHEMBL2355330 0.71 MAPT (0.78) CYP2D6CYP1A2CYP3A4CYP2C19GFER
Trifluoroacetic Acid SCHEMBL15568005 0.71 HRH1 (0.58) CYP2D6TP53KMT2AHRH1KCNH2
SCHEMBL15568738 0.71 HRH1 (0.54) CYP2D6TP53HTTALDH1A1KMT2A
SCHEMBL12811672 0.71 SOS1 (0.60) CYP2D6ALDH1A1KMT2AHRH1MEN1
SCHEMBL15569146 0.70 HRH1 (0.56) CYP2D6HTTALDH1A1KMT2AHRH1
Trifluoroacetic Acid SCHEMBL15568739 0.70 HRH1 (0.59) CYP2D6TP53HTTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed