SCHEMBL15567362

SCHEMBL15567362

CN(CCCNC(=O)C1CCN(c2nc3ccccc3n2Cc2ccc(F)cc2)CC1)C1CCCCC1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 17/20 0.69
CYP2D6 P10635 15/20 0.69
KCNH2 Q12809 8/20 0.69
CHRM1 P11229 8/20 0.66
ADRA2A P08913 1/20 0.52
HTR2B P41595 1/20 0.52
PDE4D Q08499 1/20 0.52
PDE3A Q14432 1/20 0.52
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
HTR3A P46098 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15452490 0.81 HRH1 (0.65) HRH1CYP2D6KCNH2CHRM1ALDH1A1
SCHEMBL15568738 0.79 HRH1 (0.54) HRH1CYP2D6KCNH2CHRM1MEN1
SCHEMBL27317913 0.78 HRH1 (0.69) HRH1CYP2D6KCNH2CHRM1HTR3A
Trifluoroacetic Acid SCHEMBL15568005 0.78 HRH1 (0.58) HRH1CYP2D6KCNH2CHRM1MEN1
Trifluoroacetic Acid SCHEMBL15568340 0.78 HRH1 (0.53) HRH1CYP2D6KCNH2CHRM1HTR3A
SCHEMBL15569146 0.77 HRH1 (0.56) HRH1CYP2D6KCNH2CHRM1MEN1
SCHEMBL10483537 0.77 HRH1 (0.80) HRH1CYP2D6KCNH2CHRM1ADRA2A
Trifluoroacetic Acid SCHEMBL15568739 0.76 HRH1 (0.59) HRH1CYP2D6KCNH2CHRM1ADRA2A
SCHEMBL15568448 0.76 HRH1 (0.59) HRH1CYP2D6KCNH2CHRM1MEN1
SCHEMBL15568002 0.76 CYP2D6 (0.60) HRH1CYP2D6KCNH2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed