SCHEMBL15568738

SCHEMBL15568738

O=C(NCCCN1CCN(c2ccccc2)CC1)C1CCN(c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 14/20 0.54
CYP2D6 P10635 13/20 0.54
CHRM1 P11229 5/20 0.54
KCNH2 Q12809 6/20 0.54
CHRM4 P08173 1/20 0.53
HTR3A P46098 1/20 0.51
MAPT P10636 2/20 0.51
THRB P10828 1/20 0.51
DRD2 P14416 1/20 0.50
DRD3 P35462 1/20 0.50
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL15567137 0.96 CHRM4 (0.51) HRH1CYP2D6CHRM1KCNH2CHRM4
Trifluoroacetic Acid SCHEMBL15568340 0.88 HRH1 (0.53) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL15569073 0.86 MAPT (0.48) HRH1CYP2D6CHRM1KCNH2CHRM4
SCHEMBL15567581 0.83 HRH1 (0.58) HRH1CYP2D6CHRM1KCNH2HTR3A
Trifluoroacetic Acid SCHEMBL15567853 0.82 HTR3A (0.50) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL15452490 0.81 HRH1 (0.65) HRH1CYP2D6CHRM1KCNH2HTR3A
Trifluoroacetic Acid SCHEMBL15567477 0.81 HRH1 (0.54) HRH1CYP2D6CHRM1KCNH2CHRM4
Trifluoroacetic Acid SCHEMBL15568005 0.81 HRH1 (0.58) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL27317913 0.79 HRH1 (0.69) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL15567362 0.79 HRH1 (0.69) HRH1CYP2D6CHRM1KCNH2HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed