SCHEMBL15568271

SCHEMBL15568271

CC(=O)N1CCC(C(=O)NC2CCN(c3nc4ccccc4n3Cc3ccccc3)CC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE6D O43924 5/20 0.56
CYP2D6 P10635 4/20 0.54
HRH1 P35367 4/20 0.54
CHRM1 P11229 2/20 0.54
HTR3A P46098 1/20 0.51
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
KCNH2 Q12809 2/20 0.48
BLM P54132 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL15567418 0.81 HRH1 (0.59) PDE6DCYP2D6HRH1CHRM1HTR3A
SCHEMBL15474498 0.80 PDE6D (0.66) PDE6DCYP2D6HRH1CHRM1HTR3A
SCHEMBL13181960 0.80 ALDH1A1 (0.57) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL1440257 0.79 PTGES (0.66) PDE6DALDH1A1MAPTHTTNPSR1
SCHEMBL15568544 0.79 CYP2D6 (0.54) PDE6DCYP2D6HRH1CHRM1ALDH1A1
SCHEMBL15568131 0.79 HRH1 (0.61) CYP2D6HRH1CHRM1HTR3AKCNH2
SCHEMBL15567387 0.78 TP53 (0.54) PDE6DALDH1A1NPSR1
SCHEMBL10337607 0.77 HRH1 (0.74) CYP2D6HRH1CHRM1HTR3AKCNH2
SCHEMBL15474687 0.76 PDE6D (0.79) PDE6DCYP2D6HRH1HTR3AALDH1A1
Trifluoroacetic Acid SCHEMBL15567810 0.76 HRH1 (0.57) PDE6DCYP2D6HRH1CHRM1HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed