SCHEMBL15568359

SCHEMBL15568359

Oc1cccc(-c2nc3ccccc3n2Cc2ccccc2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.76
ALDH1A1 P00352 4/20 0.74
PDE6D O43924 2/20 0.74
ALDH2 P05091 1/20 0.74
ALDH3A1 P30838 1/20 0.74
MAPT P10636 3/20 0.70
CASR P41180 1/20 0.61
HDAC1 Q13547 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
LMNA P02545 1/20 0.59
HPGD P15428 1/20 0.57
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
BRD4 O60885 4/20 0.55
TNF P01375 1/20 0.55
KDM4E B2RXH2 2/20 0.54
GAA P10253 1/20 0.54
CFTR P13569 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8021395 0.87 TP53 (0.77) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL29412044 0.86 TP53 (1.00) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL229828 0.85 ALDH1A1 (1.00) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL29412062 0.85 TP53 (0.78) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL15474496 0.85 ALDH1A1 (0.80) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL15568102 0.84 TP53 (0.76) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL11525289 0.83 KDM4E (0.59) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL6475293 0.83 ALDH1A1 (0.68) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL8025467 0.83 TP53 (0.74) TP53ALDH1A1PDE6DALDH2ALDH3A1
SCHEMBL15568695 0.83 TP53 (0.70) TP53ALDH1A1PDE6DALDH2ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed