SCHEMBL15577281

SCHEMBL15577281

CCOC(=O)C(C#N)C1(c2ccc(F)cc2)CCOC(C)(C)C1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.38
ICMT O60725 4/20 0.38
OPRM1 P35372 2/20 0.38
ALDH1A1 P00352 3/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31731178 0.89 ALDH1A1 (0.47) GAAL3MBTL1ICMTOPRM1ALDH1A1
SCHEMBL31731479 0.88 GAA (0.42) GAAL3MBTL1ICMTHTTMEN1
SCHEMBL15577185 0.88 GAA (0.44) GAAL3MBTL1ICMTTSHRMAPT
SCHEMBL31731594 0.87 ICMT (0.41) GAAL3MBTL1ICMT
SCHEMBL18112397 0.85 OPRM1 (0.41) GAAOPRM1ALDH1A1HTTMAPT
SCHEMBL627890 0.82 OPRM1 (0.43) GAAOPRM1ALDH1A1HTTMAPT
SCHEMBL12542222 0.80 OPRM1 (0.40) GAAICMTOPRM1ALDH1A1TSHR
SCHEMBL12542588 0.77 OPRM1 (0.40) OPRM1ALDH1A1TSHRMAPTSMN1; SMN2
SCHEMBL20902327 0.76 OPRM1 (0.39) GAAL3MBTL1OPRM1HTTMAPT
SCHEMBL12540893 0.76 OPRM1 (0.39) OPRM1ALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014041349-A1 TETRAHYDROPYRAN-4-YLETHYLAMINO- OR TETRAHYDROPYRANYL-4-ETHYLOXY-PYRIMIDINES OR -PYRIDAZINES AS ISOPRENYLCYSTEINCARBOXYMETHYL TRANSFERASE INHIBITORS CANCER THERAPEUTICS CRC PTY LTD (AU) 2014-03-20 WO disclosed
WO-2014041349-A1 TETRAHYDROPYRAN-4-YLETHYLAMINO- OR TETRAHYDROPYRANYL-4-ETHYLOXY-PYRIMIDINES OR -PYRIDAZINES AS ISOPRENYLCYSTEINCARBOXYMETHYL TRANSFERASE INHIBITORS CANCER THERAPEUTICS CRC PTY LTD (AU) 2014-03-20 WO disclosed