SCHEMBL15577692

SCHEMBL15577692

NC(=O)[C@H](Cc1ccc(F)cc1)Nc1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
GAA P10253 2/20 0.45
MAPK1 P28482 1/20 0.45
CA2 P00918 1/20 0.43
CA12 O43570 1/20 0.42
MMP2 P08253 1/20 0.42
ACE P12821 1/20 0.42
FOLH1 Q04609 1/20 0.41
KMT2A Q03164 2/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
SCN9A Q15858 1/20 0.41
FCER2 P06734 2/20 0.40
MMP3 P08254 1/20 0.40
MMP9 P14780 1/20 0.40
EPHX1 P07099 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521922 0.88 GPR142 (0.47) KMT2ACYP3A4CYP2C19SCN9A
SCHEMBL4523467 0.88 GPR142 (0.47) KMT2ACYP3A4CYP2C19SCN9A
SCHEMBL27723699 0.88 GPR142 (0.47) KMT2ACYP3A4CYP2C19SCN9A
SCHEMBL9169350 0.81 ALDH1A1 (0.47) ALDH1A1GAACA2CA12MMP2
SCHEMBL4528426 0.81 SCN9A (0.46) KMT2ASCN9A
SCHEMBL27723710 0.81 SCN9A (0.46) KMT2ASCN9A
SCHEMBL2722699 0.79 ELANE (0.53) FCER2EPHX1
SCHEMBL1053745 0.79 ELANE (0.53) FCER2EPHX1
SCHEMBL27746696 0.79 ALDH1A1 (0.59) ALDH1A1
SCHEMBL27509445 0.79 ALDH1A1 (0.59) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2895482-A1 HIV PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-07-22 EP claimed
WO-2014043019-A1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-03-20 WO claimed