SCHEMBL15580737

SCHEMBL15580737

C=Cc1cc(Oc2cc(Cl)c(C(=O)OC)cn2)ccc1[C@@H](C)[C@@](O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.33
SYK P43405 2/20 0.32
GPR55 Q9Y2T6 1/20 0.32
P2RX3 P56373 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
MAPT P10636 1/20 0.30
SCN9A Q15858 3/20 0.30
SCN10A Q9Y5Y9 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12164250 0.92 MALT1 (0.35) MALT1SYKGPR55P2RX3KDM4E
SCHEMBL474539 0.92 MALT1 (0.35) MALT1SYKGPR55P2RX3KDM4E
SCHEMBL2817510 0.86 MAPT (0.41) MALT1SYKGPR55KDM4ENPC1
SCHEMBL15580679 0.85 ALDH1A1 (0.32) ALDH1A1
SCHEMBL474532 0.85 GPR55 (0.33) MALT1SYKGPR55P2RX3ALDH1A1
SCHEMBL12164254 0.85 GPR55 (0.33) MALT1SYKGPR55P2RX3ALDH1A1
SCHEMBL474353 0.83 LMNA (0.41) MALT1GPR55P2RX3SCN9ASCN10A
SCHEMBL12164239 0.83 LMNA (0.41) MALT1GPR55P2RX3SCN9ASCN10A
SCHEMBL474506 0.83 ALDH1A1 (0.32) MALT1GPR55KDM4EALDH1A1MAPK1
SCHEMBL2816930 0.83 ALDH1A1 (0.32) MALT1GPR55KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed