SCHEMBL15599217

SCHEMBL15599217

Cc1cnc(OCCF)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.38
HTR2A P28223 3/20 0.35
HTR2C P28335 3/20 0.35
CYP17A1 P05093 1/20 0.34
LMNA P02545 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
APEX1 P27695 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
DRD1 P21728 1/20 0.33
KCNJ5 P48544 3/20 0.33
KCNJ3 P48549 3/20 0.33
LRRK2 Q5S007 1/20 0.32
MAPT P10636 1/20 0.32
SCN9A Q15858 1/20 0.32
APP P05067 5/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12037985 0.84 SSTR4 (0.39) SSTR4LMNACYP2C9TSHRAPEX1
SCHEMBL19823762 0.82 KCNJ5 (0.41) SSTR4CYP17A1LMNACYP2C9TSHR
SCHEMBL17248006 0.81 NOS3 (0.41) SSTR4MAPTAPP
SCHEMBL22484223 0.80 HSP90AA1 (0.41) SSTR4CYP2C9SMN1; SMN2SCN9A
SCHEMBL17815703 0.80 SSTR4 (0.38) SSTR4LMNACYP2C9TSHRAPEX1
SCHEMBL12037978 0.79 SLC13A5 (0.40) SSTR4LMNACYP2C9TSHRAPEX1
SCHEMBL15599248 0.79 CSNK2A1 (0.34) HTR2AHTR2CCYP17A1LMNACYP2C9
SCHEMBL15599195 0.78 IDH1 (0.33) HTR2AHTR2CCYP17A1CYP11B1CYP11B2
SCHEMBL15599216 0.77 SCN9A (0.44) SSTR4CYP17A1LMNACYP2C9TSHR
SCHEMBL17428846 0.77 SSTR4 (0.45) SSTR4SMN1; SMN2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970156-B1 SUBSTITUTED BENZOXAZOLES AND METHODS OF USE THEREOF GENENTECH INC (US) 2018-07-25 EP disclosed
WO-2014153037-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-09-25 WO disclosed
WO-2014144545-A2 SUBSTITUTED BENZOXAZOLES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-09-18 WO disclosed
WO-2014008458-A2 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-01-09 WO disclosed