SCHEMBL15599252

SCHEMBL15599252

CCc1cnc(CF)c(Cl)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CPB2 Q96IY4 1/20 0.31
PARP1 P09874 1/20 0.30
ALDH1A1 P00352 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20403817 0.76 CCR1 (0.34) TDP1L3MBTL1
SCHEMBL8272903 0.75 ALDH1A1 (0.44) TDP1L3MBTL1PARP1ALDH1A1NPSR1
SCHEMBL4175060 0.74 S1PR4 (0.34) CPB2ALDH1A1NPSR1
SCHEMBL19788237 0.74 CHRNB2 (0.40) TDP1L3MBTL1PARP1ALDH1A1NPSR1
SCHEMBL336025 0.73 RECQL (0.37) CPB2
SCHEMBL15220986 0.73 LOX (0.33) TDP1L3MBTL1CPB2
SCHEMBL18266782 0.73 CSNK2A1 (0.41) CPB2
SCHEMBL17002597 0.73 CPB2 (0.33) CPB2
SCHEMBL10780675 0.72 CPB2 (0.47) CPB2PARP1
SCHEMBL21120992 0.72 MRGPRX4 (0.33) RXRAGRIN1GRIN2BTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014153037-A1 SUBSTITUTED TRIAZOLOPYRIDINES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-09-25 WO disclosed
WO-2014144545-A2 SUBSTITUTED BENZOXAZOLES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-09-18 WO disclosed
WO-2014008458-A2 N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2014-01-09 WO disclosed