SCHEMBL15599982

SCHEMBL15599982

CCc1cccc2c(C(F)(F)F)c(O[C@H]3CC[C@@H](C(F)(F)F)CC3)ccc12

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 15/20 0.47
LPAR1 Q92633 1/20 0.43
AKR1B10 O60218 1/20 0.34
AKR1A1 P14550 1/20 0.34
AKR1B1 P15121 1/20 0.34
EPHX2 P34913 1/20 0.33
S1PR5 Q9H228 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15565364 0.89 ENPP2 (0.48) ENPP2LPAR1AKR1B10AKR1A1AKR1B1
SCHEMBL15599971 0.89 ENPP2 (0.48) ENPP2LPAR1AKR1B10AKR1A1AKR1B1
SCHEMBL15599984 0.85 ENPP2 (0.43) ENPP2LPAR1
SCHEMBL20403951 0.84 ENPP2 (0.45) ENPP2LPAR1S1PR5
SCHEMBL15600021 0.83 ENPP2 (0.48) ENPP2LPAR1EPHX2S1PR5
SCHEMBL15564597 0.83 ENPP2 (0.48) ENPP2LPAR1EPHX2S1PR5
SCHEMBL15599979 0.83 ENPP2 (0.49) ENPP2LPAR1AKR1B10AKR1A1AKR1B1
SCHEMBL20403997 0.83 ENPP2 (0.49) ENPP2LPAR1AKR1B10AKR1A1AKR1B1
SCHEMBL20403979 0.82 ENPP2 (0.52) ENPP2LPAR1S1PR5
SCHEMBL15599983 0.82 ENPP2 (0.57) ENPP2LPAR1AKR1B10AKR1A1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014025709-A1 COMPOUNDS THAT ARE S1P MODULATING AGENTS AND/OR ATX MODULATING AGENTS BIOGEN IDEC MA INC. (US) 2014-02-13 WO disclosed