SCHEMBL15638569

SCHEMBL15638569

O=C(N=C(c1ccccc1)c1ccccc1)c1ccccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.59
AGTR1 P30556 3/20 0.58
LMNA P02545 5/20 0.55
NAPRT Q6XQN6 1/20 0.55
P4HTM Q9NXG6 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
KDM4E B2RXH2 5/20 0.51
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
PKM P14618 2/20 0.50
MITF O75030 2/20 0.50
CDK5 Q00535 1/20 0.50
CDK5R1 Q15078 1/20 0.50
NCOA1 Q15788 1/20 0.49
NCOA3 Q9Y6Q9 1/20 0.49
ALDH1A1 P00352 4/20 0.48
MAPT P10636 4/20 0.47
HPGD P15428 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13127271 0.78 CES2 (0.55) KMT2ALMNANAPRTP4HTML3MBTL1
SCHEMBL2006799 0.77 CES2 (0.64) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL28250849 0.76 CES1 (0.48) KMT2ALMNANAPRTL3MBTL1CES2
SCHEMBL322444 0.76 AGTR1 (0.58) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL3777401 0.76 LMNA (0.61) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL11768655 0.76 AGTR1 (0.58) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL29498791 0.76 AGTR1 (0.58) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL322443 0.76 AGTR1 (0.58) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL398165 0.75 KMT2A (1.00) KMT2AAGTR1LMNANAPRTP4HTM
SCHEMBL29373829 0.75 KMT2A (1.00) KMT2AAGTR1LMNANAPRTP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903989-A1 PYRROLO[2,3-D]PYRIMIDINE TROPOMYOSIN-RELATED KINASE INHIBITORS Pfizer Limited (GB) 2015-08-12 EP disclosed
WO-2014053967-A1 PYRROLO[2,3-D]PYRIMIDINE TROPOMYOSIN-RELATED KINASE INHIBITORS PFIZER LIMITED (GB) 2014-04-10 WO disclosed