SCHEMBL15664381

SCHEMBL15664381

Cc1csc(NC(=O)Oc2nc(C)ccc2Nc2cccnc2C)n1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.42
RAB9A P51151 7/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 3/20 0.41
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40
ALDH1A1 P00352 3/20 0.40
POLB P06746 3/20 0.40
MAPK1 P28482 2/20 0.40
GRM5 P41594 1/20 0.40
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HTT P42858 2/20 0.39
TP53 P04637 1/20 0.39
RCE1 Q9Y256 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15663530 0.83 RAB9A (0.52) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL15663528 0.82 GRM5 (0.48) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL15663516 0.81 MAPT (0.46) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL15663466 0.80 SMARCA2 (0.42) NPC1RAB9ASMARCA2SMARCA4POLB
SCHEMBL15663669 0.79 GRM5 (0.44) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL15664200 0.78 LPAR1 (0.34) NPC1RAB9AMAPTGRM5HTT
SCHEMBL15663616 0.78 MAPT (0.40) NPC1RAB9ASMN1; SMN2HPGDMAPT
SCHEMBL15664001 0.78 PDE4B (0.40) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL15663526 0.78 GRM5 (0.40) GRM5
SCHEMBL15663949 0.76 RAB9A (0.41) NPC1RAB9ASMN1; SMN2HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858854-B1 PYRIDINE-2-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-05-07 EP claimed