SCHEMBL15670499

SCHEMBL15670499

CON(C)C(=O)CN(C(=O)OC(C)(C)C)c1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KCNQ4 P56696 3/20 0.34
KCNQ5 Q9NR82 3/20 0.34
MLYCD O95822 2/20 0.34
LMNA P02545 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRM1 P35372 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
POLQ O75417 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14830095 0.87 MT-CO2 (0.44) NPSR1HSD17B10MEN1KMT2A
SCHEMBL3349318 0.82 MLYCD (0.41) KCNQ4KCNQ5MLYCDLTB4R2MEN1
SCHEMBL2900197 0.80 KDM1A (0.42) KDM1AHDAC8HDAC6KCNQ4KCNQ5
SCHEMBL8289776 0.78 F2 (0.38) KCNQ4KCNQ5MEN1KMT2A
SCHEMBL8349153 0.76 SSTR4 (0.43) KCNQ4KCNQ5MLYCDLMNANPSR1
SCHEMBL9222980 0.75 KCNQ4 (0.41) KDM1AHDAC8HDAC6KCNQ4KCNQ5
SCHEMBL24232684 0.74 POLQ (0.42) KCNQ4KCNQ5LMNAHSD17B10POLQ
SCHEMBL4664640 0.73 SMN1; SMN2 (0.45) L3MBTL1NPSR1MEN1KMT2AOPRM1
SCHEMBL3989317 0.73 KMT2A (0.35) KDM1AHDAC8HDAC6KCNQ4KCNQ5
SCHEMBL6217029 0.73 MAPT (0.36) KCNQ4KCNQ5MLYCDLMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2912034-A1 3,4-DISUBSTITUTED OXAZOLIDINONE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE CALCIUM ACTIVATED POTASSIUM CHANNEL F. Hoffmann-La Roche AG (CH) 2015-09-02 EP disclosed
WO-2014067861-A1 3,4-DISUBSTITUTED OXAZOLIDINONE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE CALCIUM ACTIVATED POTASSIUM CHANNEL F. HOFFMANN-LA ROCHE AG (CH) 2014-05-08 WO disclosed