SCHEMBL15701166

SCHEMBL15701166

CC(C(=O)Nc1ccc2nc(NC(=O)c3cscn3)sc2c1)c1cccc(CF)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 13/20 0.46
NPC1 O15118 9/20 0.46
CASP3 P42574 2/20 0.45
SENP8 Q96LD8 2/20 0.45
SENP7 Q9BQF6 2/20 0.45
SENP6 Q9GZR1 2/20 0.45
KDM4E B2RXH2 7/20 0.44
POLB P06746 4/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 1/20 0.44
MAPT P10636 10/20 0.42
OPRK1 P41145 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HTT P42858 2/20 0.42
PKM P14618 2/20 0.42
AGTR1 P30556 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
KMT2A Q03164 4/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15701057 0.90 CASP3 (0.45) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701165 0.88 ACP1 (0.46) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL19446717 0.88 RAB9A (0.52) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701244 0.87 CYP2C9 (0.49) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701145 0.85 PSEN1 (0.46) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701026 0.85 RAB9A (0.48) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701278 0.84 CASP3 (0.50) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701115 0.84 MAPT (0.51) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701087 0.84 CYP2C9 (0.51) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL15701093 0.84 CYP2C9 (0.51) RAB9ANPC1CASP3SENP8SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014070979-A1 INHIBITORS OF CYTOMEGALOVIRUS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-05-08 WO disclosed