SCHEMBL15701635

SCHEMBL15701635

NS(=O)(=O)c1ccc2c(ccn2Cc2cccc(Cl)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.39
AURKA O14965 1/20 0.39
DCLK1 O15075 1/20 0.39
PDPK1 O15530 1/20 0.39
JAK2 O60674 1/20 0.39
ROCK2 O75116 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
EGFR P00533 1/20 0.39
NTRK1 P04629 1/20 0.39
PRKCG P05129 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
CDK1 P06493 1/20 0.39
LYN P07948 1/20 0.39
RET P07949 1/20 0.39
IGF1R P08069 1/20 0.39
ROS1 P08922 1/20 0.39
FGFR1 P11362 1/20 0.39
SRC P12931 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14149420 0.75 CA12 (0.52) NR1I2PLA2G4ACA1CA2CA9
SCHEMBL14061517 0.73 ALDH1A1 (0.53) PLA2G4ALMNA
SCHEMBL14061528 0.72 CA1 (0.41) PLA2G4ACA1CA2CA9LMNA
SCHEMBL10179526 0.71 PTGS2 (0.37) NR1I2NPC1HSP90AA1KMT2A
SCHEMBL14058826 0.71 ROCK1 (0.45) CA1CA2CA4CA9NPC1
SCHEMBL14141758 0.70 KMT2A (0.39) NR1I2KMT2A
SCHEMBL19476152 0.66 NPC1 (0.54) NR1I2NPC1HSP90AA1
SCHEMBL14061276 0.65 LMNA (0.47) PLA2G4ACA1CA2CA4CA9
SCHEMBL8761290 0.65 PRKCI (0.55) CA1CA2CA9LMNACA12
SCHEMBL1243312 0.65 POLB (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140135318-A1 SUBSTITUTED SULFONAMIDES USEFUL AS ANTIAPOPTOTIC BCL INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2014-05-15 US disclosed
US-20140135318-A1 SUBSTITUTED SULFONAMIDES USEFUL AS ANTIAPOPTOTIC BCL INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2014-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140135318-A1 SUBSTITUTED SULFONAMIDES USEFUL AS ANTIAPOPTOTIC BCL INHIBITORS BCL2, BAX, BCL2A1 NR1I2 2401/4885AURKA 4211/4885DCLK1 3616/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.