SCHEMBL1570170

SCHEMBL1570170

N#CC(SC(F)(F)F)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
TRPA1 O75762 1/20 0.42
ALDH1A1 P00352 5/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
USP2 O75604 1/20 0.33
MAP2K1 Q02750 1/20 0.33
AR P10275 2/20 0.33
TNF P01375 1/20 0.32
NOD2 Q9HC29 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
NOD1 Q9Y239 1/20 0.32
CTSL P07711 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
LRRK2 Q5S007 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28321971 0.80 TRPA1 (0.42) TSHRTRPA1ALDH1A1MAPTHTT
SCHEMBL11099247 0.80 ALDH1A1 (0.30) ALDH1A1MAPT
SCHEMBL28515424 0.76 TSHR (0.50) TSHRTRPA1ALDH1A1MAPTHTT
SCHEMBL9493266 0.72 TSHR (0.46) TSHRTRPA1ALDH1A1MAPTHTT
SCHEMBL28929083 0.72 TSHR (0.46) TSHRTRPA1ALDH1A1MAPTHTT
SCHEMBL22190304 0.72 TSHR (0.40) TSHRALDH1A1TAAR1DPP4
SCHEMBL28518519 0.71 PTGS2 (0.37) TSHRTRPA1ALDH1A1MAPTCTSL
SCHEMBL1021030 0.68 TSHR (0.46) TSHRTRPA1ALDH1A1MAPTHTT
SCHEMBL2155150 0.68 TSHR (0.44) TSHRALDH1A1TAAR1DPP4
SCHEMBL31130672 0.68 SRC (0.39) TSHRLMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307397-A1 6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACID DERIVATIVES Array Biopharma, Inc. (US) 2011-04-13 EP disclosed
WO-2009158426-A1 6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2009-12-30 WO disclosed
EP-0066482-B1 METHOD FOR THE PREPARATION OF ALIPHATIC OR AROMATIC NITRILES RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1984-11-28 EP disclosed
EP-0065447-B1 FLUOR-CONTAINING SILICA CATALYSTS; THEIR PREPARATION, AND THEIR USE IN THE PREPARATION OF NITRILES RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1984-09-05 EP disclosed
EP-0066482-A1 Method for the preparation of aliphatic or aromatic nitriles RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1982-12-08 EP disclosed
EP-0066483-A1 Method for the preparation of aliphatic or aromatic nitriles RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1982-12-08 EP disclosed
EP-0065447-A1 Fluor-containing silica catalysts; their preparation, and their use in the preparation of nitriles RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1982-11-24 EP disclosed