SCHEMBL15713614

SCHEMBL15713614

C=C(O)c1ccc(NS(=O)(=O)c2cccc3cccnc23)cc1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.72
GAA P10253 2/20 0.72
MEN1 O00255 4/20 0.68
KMT2A Q03164 4/20 0.68
TP53 P04637 1/20 0.64
HTT P42858 1/20 0.64
PKM P14618 1/20 0.62
PKLR P30613 7/20 0.60
HDAC1 Q13547 1/20 0.60
GFER P55789 1/20 0.59
FABP1 P07148 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2702246 0.88 ALDH1A1 (0.76) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL30708093 0.88 ALDH1A1 (0.76) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL18753536 0.85 ALDH1A1 (0.78) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL808364 0.84 ALDH1A1 (1.00) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL15480551 0.84 MEN1 (0.73) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL17210223 0.82 ALDH1A1 (1.00) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL10192086 0.81 MEN1 (0.75) ALDH1A1GAAMEN1KMT2ATP53
SCHEMBL22394150 0.81 PKLR (0.82) PKMPKLR
SCHEMBL2702840 0.80 PKLR (0.79) PKMPKLR
SCHEMBL3555597 0.80 FABP1 (0.74) ALDH1A1GAAMEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014074848-A1 THERAPEUTIC COMPOUNDS AND COMPOSITIONS AND THEIR USE AS PKM2 MODULATORS AGIOS PHARMACEUTICALS, INC. (US) 2014-05-15 WO disclosed