SCHEMBL15718288

SCHEMBL15718288

CNC(=O)c1ccn2nccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.47
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
NTRK1 P04629 1/20 0.44
ADRA1A P35348 2/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
ADRA1D P25100 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1B P35368 1/20 0.44
DRD3 P35462 1/20 0.44
HTR2B P41595 1/20 0.44
PLK1 P53350 1/20 0.44
ESR1 P03372 1/20 0.44
FASN P49327 1/20 0.43
RIPK1 Q13546 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30980395 0.84 AOC2 (0.50) NAMPTNTRK1ADRA1AHTR1ADRD2
SCHEMBL2176055 0.81 ESR1 (0.46) NAMPTNTRK1ADRA1AHTR1ADRD2
SCHEMBL3642134 0.81 JMJD6 (0.44) NAMPTADRA1AHTR1ADRD2DRD1
SCHEMBL3081703 0.80 ESR1 (0.47) NAMPTADRA1AHTR1ADRD2DRD1
SCHEMBL15718194 0.79 RAB9A (0.51) NAMPTADRA1AHTR1ADRD2DRD1
SCHEMBL3089155 0.78 ESR1 (0.43) NAMPTNTRK1ADRA1AHTR1ADRD2
SCHEMBL27906136 0.77 ESR1 (0.52) NAMPTNTRK1ADRA1AHTR1ADRD2
SCHEMBL27326899 0.77 ALDH1A1 (0.44) HDAC8HDAC6PLK1THRBHDAC2
SCHEMBL31288941 0.77 MAPK1 (0.52) NAMPTNTRK1TDP1
SCHEMBL31205259 0.77 ESR1 (0.45) NAMPTNTRK1ADRA1AHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4695248-A1 PYRAZOLO[1,5-A]PYRIDINE DERIVATIVES Syngenta Crop Protection AG (CH) 2026-02-18 EP disclosed
WO-2024213663-A1 PYRAZOLO[1,5-A]PYRIDINE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2024-10-17 WO disclosed
EP-2925757-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES Novartis AG (CH) 2015-10-07 EP disclosed
WO-2014078802-A1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES IRM LLC (BM) 2014-05-22 WO disclosed