SCHEMBL1574577

SCHEMBL1574577

CC(=O)c1sc(-c2cccnc2)nc1C

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.77
CYP1A2 P05177 4/20 0.77
CYP2C19 P33261 4/20 0.77
LMNA P02545 1/20 0.77
KMT2A Q03164 4/20 0.62
MEN1 O00255 3/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2D6 P10635 1/20 0.62
MAPT P10636 2/20 0.59
RAB9A P51151 1/20 0.58
ALDH1A1 P00352 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
KDM4E B2RXH2 2/20 0.55
CYP2A6 P11509 1/20 0.52
NT5E P21589 1/20 0.52
BRAF P15056 1/20 0.52
HPGD P15428 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CDC7 O00311 2/20 0.51
DBF4 Q9UBU7 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29783018 1.00 CYP3A4 (0.77) CYP3A4CYP1A2CYP2C19LMNAKMT2A
Hydrochloric Acid SCHEMBL1679765 0.99 CYP3A4 (0.75) CYP3A4CYP1A2CYP2C19LMNAKMT2A
SCHEMBL289321 0.89 CYP3A4 (0.62) CYP3A4CYP1A2CYP2C19LMNAKMT2A
SCHEMBL11387955 0.89 CYP1A2 (0.73) CYP3A4CYP1A2CYP2C19LMNAKMT2A
SCHEMBL595294 0.88 CYP1A2 (0.77) CYP3A4CYP1A2CYP2C19LMNAKMT2A
Hydrochloric Acid SCHEMBL289747 0.88 CYP3A4 (0.61) CYP3A4CYP1A2CYP2C19LMNAKMT2A
SCHEMBL5211666 0.87 CYP1A2 (1.00) CYP3A4CYP1A2CYP2C19LMNAKMT2A
Hydrochloric Acid SCHEMBL11388179 0.87 CYP1A2 (0.75) CYP3A4CYP1A2CYP2C19LMNAKMT2A
SCHEMBL3065347 0.87 CYP1A2 (0.75) CYP3A4CYP1A2CYP2C19LMNAKMT2A
Hydrochloric Acid SCHEMBL11388173 0.86 CYP1A2 (0.73) CYP3A4CYP1A2CYP2C19LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114990587-B Electrochemical synthesis method of thiazole compound 华南理工大学 2023-05-23 CN disclosed
CN-114990587-A Electrochemical synthesis method of thiazole compound 华南理工大学 2022-09-02 CN disclosed
EP-3954681-A1 SPIROHEPTANE SALICYLAMIDES AND RELATED COMPOUNDS AS INHIBITORS OF ROCK Bristol-Myers Squibb Company (US) 2022-02-16 EP disclosed
EP-3402790-B1 SPIROHEPTANE SALICYLAMIDES AND RELATED COMPOUNDS AS INHIBITORS OF ROCK BRISTOL MYERS SQUIBB CO (US) 2021-10-06 EP disclosed
US-9451775-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-09-27 US disclosed
US-9451775-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-09-27 US disclosed
US-9451775-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-09-27 US disclosed
EP-2583556-B1 Heterocyclic compounds as pest controllers BAYER CROPSCIENCE AG (DE) 2016-01-20 EP disclosed
EP-2583556-B1 Heterocyclic compounds as pest controllers BAYER CROPSCIENCE AG (DE) 2016-01-20 EP disclosed
EP-2591674-B1 Heterocyclic compounds as pest controllers BAYER CROPSCIENCE AG (DE) 2016-01-13 EP disclosed
EP-1581231-A1 ANTI-VIRAL COMPOUNDS Cyclacel Limited (GB) 2005-10-05 EP disclosed
WO-2004043467-A1 ANTI-VIRAL COMPOUNDS CYCLACEL LIMITED (GB) 2004-05-27 WO disclosed
US-6699854-B2 2-SUBSTITUTED 4-HETEROARYL- PYRIMIDINES, INHIBITORS OF CYCLIN-DEPENDENT KINASES (CDKS) CYCLACEL LIMITED (GB) 2004-03-02 US disclosed
US-20030149057-A1 Anti-cancer compounds CYCLACEL LIMITED (GB) 2003-08-07 US disclosed
CN-1420884-A 2-substituted 4-heteroaryl-pyrimidines and their use in the treatment of proliferative diseases CYCLACEL LTD (GB) 2003-05-28 CN disclosed
US-6531479-B2 Anticancer agents, skin disorders CYCLACEL LIMITED (GB) 2003-03-11 US disclosed
EP-1274705-A1 2-SUBSTITUTED 4-HETEROARYL-PYRIMIDINES AND THEIR USE IN THE TREATMENT OF PROLIFERATIVE DISORDERS Cyclacel Limited (GB) 2003-01-15 EP disclosed
US-20020019404-A1 Anti-cancer compounds CYCLACEL LIMITED (GB) 2002-02-14 US disclosed
WO-2001072745-A1 2-SUBSTITUTED 4-HETEROARYL-PYRIMIDINES AND THEIR USE IN THE TREATMETN OF PROLIFERATIVE DISORDERS CYCLACEL LIMITED (GB) 2001-10-04 WO disclosed
US-4080457-A INSECTICIDES, PESTICIDES, MITICIDES UNIROYAL CHEMICAL COMPANY, INC. 1978-03-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019404-A1 Anti-cancer compounds CDK3, CDK2, CDK4 CYP3A4 2674/4885CYP1A2 2580/4885CYP2C19 2882/4885
US-20030149057-A1 Anti-cancer compounds CDK3, CDK2, CDK4 CYP3A4 2674/4885CYP1A2 2580/4885CYP2C19 2882/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.