SCHEMBL15760955

SCHEMBL15760955

CCc1nc(NC)c2c(=O)[nH]cnc2n1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
XDH P47989 5/20 0.39
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 1/20 0.36
PDPK1 O15530 2/20 0.34
TMIGD3 P0DMS9 1/20 0.34
CYP2C9 P11712 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
DYRK1A Q13627 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15760951 0.80 XDH (0.62) XDHALDH1A1TMIGD3KDM4EPARP1
SCHEMBL15803493 0.78 CYP1A2 (0.45) XDHALDH1A1CYP1A2CYP2D6PDPK1
SCHEMBL16146652 0.78 XDH (0.63) XDHCYP1A2CYP2D6HTT
SCHEMBL15760953 0.75 PDPK1 (0.39) XDHALDH1A1CYP1A2CYP2D6PDPK1
SCHEMBL15803489 0.75 JAK2 (0.41)
SCHEMBL15760947 0.74 PARP1 (0.38) XDHCYP1A2CYP2D6PDPK1TMIGD3
SCHEMBL16146651 0.71 XDH (0.39) XDHALDH1A1PDPK1KDM4EGAA
SCHEMBL26175667 0.67 XDH (0.50) XDHCYP1A2CYP2D6CYP2C9
SCHEMBL10408919 0.67 ADORA3 (0.50) XDHCYP1A2CYP2D6TMIGD3HTT
SCHEMBL15760952 0.67 PARP1 (0.43) XDHALDH1A1PDPK1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140171429-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-19 US disclosed
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140171429-A1 BICYCLIC INHIBITORS OF ALK ALK, ACVR1, ACVR1B XDH 1213/4885ALDH1A1 161/4885CYP1A2 751/4885
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ALK, ABL1, BOD1L1 XDH 603/4885ALDH1A1 140/4885CYP1A2 824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.