SCHEMBL157686

SCHEMBL157686

[c]1nc(-c2ccon2)co1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CHRM1 P11229 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3082762 0.76 NPC1 (0.42) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL1126619 0.68
Methoxymethane SCHEMBL27908243 0.67 RAB9A (0.50) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL7387155 0.67 ALDH1A1 (0.35) CYP1A2CYP2D6CYP2C19
SCHEMBL28934089 0.66
SCHEMBL970674 0.65 KDM4E (0.56) CYP1A2CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL2675050 0.65 KDM4E (0.43) CYP19A1NPC1RAB9AKDM4E
SCHEMBL718110 0.65 CYP1A2 (0.34) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL1638199 0.65 CYP1A2 (0.34) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL27774669 0.65 NPC1 (0.33) CYP1A2CYP2D6CYP19A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 121 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101466678-B Substituted 3-cyanopyridines as protein kinase inhibitors WYETH CORP 2012-12-26 CN claimed
CN-102485743-A Antineoplastic compound BEIJING HANMEI PHARMACEUTICAL CO LTD 2012-06-06 CN claimed
CN-101779124-A modulation of chemosensory receptors and ligands associated therewith SENOMYX INC 2010-07-14 CN claimed
US-20070259879-A1 Piperazine and piperidine biaryl derivatives TRIMERIS, INC. 2007-11-08 US claimed
CN-1802348-A Mercapto-phenyl-naphthyl-methane derivatives and preparation thereof COUNCIL SCIENT IND RES (IN) 2006-07-12 CN claimed
CN-1688578-A Phosphodiesterase 4 inhibitors MEMORY PHARM CORP (US) 2005-10-26 CN claimed
WO-2005037797-A1 SUBSTITUTED PYRAZOLE UREA COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2005-04-28 WO claimed
CN-1578660-A Lactam-containing compounds and derivatives thereof as factor xa inhibitors BRISTOL MYERS SQUIBB CO (US) 2005-02-09 CN claimed
EP-0983272-B1 A NEW CLASS OF BENZOPORPHYRIN DERIVATIVE PHOTOACTIVE COMPOUNDS UNIV BRITISH COLUMBIA (CA) 2003-10-29 EP claimed
CN-1120166-C New class of benzoporphyrin derivative photoactive compounds UNIV BRITISH COLUMBIA (CA) 2003-09-03 CN claimed
CN-1255135-A New class of benzoporphyrin derivative photoactive compounds UNIV BRITISH COLUMBIA (CA) 2000-05-31 CN claimed
CN-1138332-A Pyridazinoquinoline compounds ZENECA LTD (GB) 1996-12-18 CN claimed
EP-3566055-A1 METHODS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS Yumanity Therapeutics, Inc. (US) 2019-11-13 EP disclosed
WO-2018129403-A1 METHODS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS YUMANITY THERAPEUTICS (US) 2018-07-12 WO disclosed
CN-103508961-B Antitumor drug CROWN BIOSCIENCE TAICANG CO LTD 2015-07-22 CN disclosed
CN-103508961-A Antitumor drug CROWN BIOSCIENCE TAICANG CO LTD 2014-01-15 CN disclosed
CN-1151400-A Novel sulfonylaminopyrimidines HOFFMANN LA ROCHE (CH) 1997-06-11 CN disclosed
CN-1138332-A Pyridazinoquinoline compounds ZENECA LTD (GB) 1996-12-18 CN disclosed
EP-0630370-A1 FUNGICIDAL OXAZOLIDINONES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1994-12-28 EP disclosed
WO-1993018016-A1 FUNGICIDAL OXAZOLIDINONES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070259879-A1 Piperazine and piperidine biaryl derivatives CYP3A5, CYP3A43, CCR5 CYP1A2 8/4885CYP2D6 31/4885CYP19A1 700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.